This drug is designed for suppression of aromatization and decreases its activity with 80-90% from its initial level. It differs from other drugs with high effectiveness and effect rate. Even after some hours of administration the aromatization process is about totally blocked thanks to the maximal concentration of the drug.
The effect mechanism of Anastrozol from Balkan Pharmaceuticals is fundamentally different from the known Tamoxifen which blocks the only estrogen but doesn’t stop the process of aromatization itself. This drug prevents only aromatization; consequently, the estrogens in the organism are not synthesized and are not produced. One-time administration of Anastrazol of 1 mg provides the decrease of estradiol production in blood by 80% within first hours after being applied.
First drugs of such type were designed practically simultaneously with Tamoxifen, in 1980s in United States. From that time by 1995 third generation of aromatase inhibitors appeared to which Anastrozole and its analogues (Arimidex) are included and their sale started. In medicine they are used at malignant neoplasm of breast, with high activity of estrogen receptors in the tumor tissue.
Designed to be used by women during the period of menopause. Since many forms of breast cancer are stimulated by estrogen, this drug is intended to decrease the quantity of estrogen in blood, slowing the development of the disease in this way. In some experimental researches the level of estradiol in the blood decrease up to 98% of the initial concentration.
In bodybuilding the active substance of the drug anastrozole is used for the prophylaxis of gynecomasty and fat accumulation, side effects due to the use of testosterone esters and other drugs with androgenic activity. It is recommended only to experienced and professional sportsmen who apply courses with the esters of testosterone, sustanon and other drugs with androgenic activity. The cost of Anastrozol (Balkan) quite justifies itself because one tablet per day is enough. Administration is started either when the course of steroids is started or when first manifestations of aromatization are observed, using 0,25-1 mg daily. It is better to apply the drug at an empty stomach because it is absorbed faster and more completely from gastrointestinal tract to the blood system. The maximum concentration in the blood is reached 2 hours after the administration.
Course of Anastrozole (Balkan Pharmaceuticals) during 10-14 days decreases the side effects coming from heavy steroids courses, for example, 200-300 mg of testosterone propionate daily. The effectiveness of the drug is also confirmed by numerous clinical tests but due to the power of its effect it is not recommended to everyone.
Detailed instruction to Anastrozole tablets is posted at our Forum where you may learn about individual recommendation on drug administration. It’s desirable to administrate the drug at an experienced specialist’s control. The drug itself has androgenic and progestogenic activity, doesn’t affect the secretion of aldosterone and cortisol, doesn’t need the injection of corticosteroids during the course.
Anastrozole has long half-life period (40-50 hours) and, even at small dosages, effectively prevents feminization manifestations at sportsmen. Excreted from the organism mainly with urine and bile. Does not affect the production of natural testosterone. Administration of more than 1 mg of the drug daily and during long period is not recommended.
Reviews about Anastrozole
With all its advantages, sportsmen distinguish two main disadvantages of the drug. Decrease of estrogen side effects are confirmed in all reviews about Anastrozole (Balkan), so that its effectiveness is quite proved. But during the process of active affect the drug suppresses also the synthesis of “good” cholesterol that is necessary for cardiovascular system, this is the first disadvantage.
Reviews about anastrozole and our Forum don’t recommend using the drug by those people who have problems with heart or vessels. Tamoxifen becomes an alternative in this case. In combination with finasteride the reviews about Anastrozole recommend using the drug for minimization of side effects of steroids that are converted to dihydrotestosterone. This affects the state of the musculature only in a positive way. After studying the reviews about Anastrozole, the second disadvantage could be named its relatively high price. The application of the drug pays off in case of long course or courses with high doses of steroids.
Even combined administration of Tamoxifen and Proviron doesn’t give the result like this drug does. That’s why quite a high price of Anastrozole is quite justified by the effectiveness of the drug. People with sensitivity to the drug may have some side effects: acne, nausea, headache, sleepiness, and allergy reactions.
Price for Anastrozole is conditioned with the expense of synthesis of the drug itself and may often be higher than the price of the steroids themselves which, naturally, doesn’t make the bodybuilders happy. But it is no worth to economize on your health. Compare what is more profitable – price for Anastrozol or numerous visits to doctors and performing surgical operations fighting agains gynecomasty.
The cost of real qualitative drug is always higher than of cheaper analogues. That is why you should keep in mind that if you see a shop where the price of Anastrozol (Balkan) is attractively low, don’t be mistaken, this is the first characteristic of fake drug. The drugs purchased in our internet shop are the production of licensed factories of sports pharmacology. So, the originality of the drug that you purchased may be checked by UPIC number that is placed at the package on producer’s official website – www.b-p.md
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